Sunepitron

{{Drugbox-lat | IUPAC_name = 1-{[2-(pirimidin-2-il)oktahidro-2H-pirido[1,2-a]pirazin-7-il]metil}pirolidin-2,5-dion | image = Sunepitron.png | width = | image2 = | width2 =

| tradename = | pregnancy_category = | legal_status = Nije kontrolisana supstanca | routes_of_administration = Oralno

| bioavailability = | metabolism = | elimination_half-life = | excretion =

| CAS_number_Ref =  ^Y | CAS_number = 148408-65-5 | ATC_prefix = none | ATC_suffix = | PubChem = 9799246 | IUPHAR_ligand = | ChEMBL_Ref = | ChemSpiderID = 7975011 | UNII_Ref =  ^Y | UNII = 2GT50C8U60 | KEGG = D02569 | ChEMBL = 380369 | DrugBank_Ref = | DrugBank =

| C=17 | H=23 | N=5 | O=2 | molecular_weight = 329,40 g/mol | smiles = O=C1N(C(=O)CC1)CC4CCC3N(CCN(c2ncccn2)C3)C4 | StdInChI_Ref =  ^Y | StdInChI = | StdInChIKey_Ref =  ^Y | StdInChIKey = }}

Sunepitron (CP-93,393) je kombinovani agonist 5-HT_1A receptora i antagonist α₂-adrenergičkog receptora. On je bio u razvoju za tretiranje depresije i anksioznosti. Dospeo je do faze III kliničkih ispitivanja pre nego što je razvoj prekinut.

Sinteza

Jedan od mogućih sintetičkih puteva je:

Vidi još

• Lezopitron

Literatura

• Kaplan, Eliot F.; Turkington, Carol (2001). Making the antidepressant decision: how to choose the right treatment option for you and your loved ones. Chicago, Ill: Contemporary Books. ISBN 978-0-7373-0417-6. 
• Stahl, S. M. (2000). Essential psychopharmacology: neuroscientific basis and practical application. Cambridge, UK: Cambridge University Press. ISBN 978-0-521-64615-4. 
• Kaplan, Eliot F.; Turkington, Carol (2001). Making the antidepressant decision: how to choose the right treatment option for you and your loved ones. Chicago, Ill: Contemporary Books. ISBN 978-0-7373-0417-6. 
• Stahl, S. M. (2000). Essential psychopharmacology: neuroscientific basis and practical application. Cambridge, UK: Cambridge University Press. ISBN 978-0-521-64615-4.